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ACS Medicinal Chemistry Letters(4,993)
ISSN: 1948-5875
1    
Identification of potent, selective, cell-Active inhibitors of the histone lysine methyltransferase EZH2 期刊论文

ACS Medicinal Chemistry Letters     ISSN:1948-5875  Volume:3  Issue:12  Page:1091-1096  

Verma Sharad K;   Tian Xinrong;   Lafrance Louis V;   Duquenne Céline;   Suarez Dominic P;   ...

来源数据库:[Web of Science, Science Citation Index Expanded, Scopus]         被引频次:181

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2    
Discovery of a potent and selective BCL-X L inhibitor with in vivo activity 期刊论文

ACS Medicinal Chemistry Letters     ISSN:1948-5875  Volume:5  Issue:10  Page:1088-1093  

Tao Zhi-Fu;   Hasvold Lisa;   Wang Le;   Wang Xilu;   Petros Andrew M;   ...

被引频次:91

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3    
Discovery of GSK2126458, a highly potent inhibitor of PI3K and the mammalian target of rapamycin 期刊论文

ACS Medicinal Chemistry Letters     ISSN:1948-5875  Volume:1  Issue:1  Page:39-43  

Knight Steven D;   Adams Nicholas D;   Burgess Joelle L;   Chaudhari Amita M;   Darcy Michael G;   ...

来源数据库:Scopus        

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4    
Discovery of RG7112: A small-molecule MDM2 inhibitor in clinical development 期刊论文

ACS Medicinal Chemistry Letters     ISSN:1948-5875  Volume:4  Issue:5  Page:466-469  

Vu Binh;   Wovkulich Peter;   Pizzolato Giacomo;   Lovey Allen;   Ding Qingjie;   ...

来源数据库:[Web of Science, Science Citation Index Expanded, Scopus]         被引频次:106

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5    
INCB24360 (Epacadostat), a Highly Potent and Selective Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitor for Immuno-oncology 期刊论文

ACS Medicinal Chemistry Letters     ISSN:1948-5875  Volume:8  Issue:5  Page:486-491  

Yue Eddy W;   Sparks Richard;   Polam Padmaja;   Modi Dilip;   Douty Brent;   ...

来源数据库:Scopus        

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6    
INCB24360 (Epacadostat), a Highly Potent and Selective Indoleamine-2,3-dioxygenase 1 (ID01) Inhibitor for Immunooncology 期刊论文

ACS MEDICINAL CHEMISTRY LETTERS     ISSN:1948-5875  Volume:8  Issue:5  Page:486-491  

Yue EW;   Sparks R;   Polam P;   Modi D;   Douty B;   ...

被引频次:46

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7    
Biocatalysis in the Pharmaceutical Industry: The Need for Speed 期刊论文

ACS Medicinal Chemistry Letters     ISSN:1948-5875  Volume:8  Issue:5  Page:476-480  

Truppo Matthew D;  

来源数据库:[Web of Science, Science Citation Index Expanded, Scopus]         被引频次:45

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8    
Discovery of the first potent inhibitors of mutant IDH1 that lower tumor 2-HG in vivo 期刊论文

ACS Medicinal Chemistry Letters     ISSN:1948-5875  Volume:3  Issue:10  Page:850-855  

Popovici-Muller Janeta;   Saunders Jeffrey O;   Salituro Francesco G;   Travins Jeremy M;   Yan Shunqi;   ...

来源数据库:[Web of Science, Science Citation Index Expanded, Scopus]         被引频次:114

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9    
Design and Synthesis of Tesirine, a Clinical Antibody-Drug Conjugate Pyrrolobenzodiazepine Dimer Payload 期刊论文

ACS Medicinal Chemistry Letters     ISSN:1948-5875  Volume:7  Issue:11  Page:983-987  

Tiberghien Arnaud C;   Levy Jean-Noel;   Masterson Luke A;   Patel Neki V;   Adams Lauren R;   ...

来源数据库:[Web of Science, Science Citation Index Expanded, Scopus]         被引频次:41

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10    
Identification of NVP-BKM120 as a potent, selective, orally bioavailable class i PI3 kinase inhibitor for treating cancer 期刊论文

ACS Medicinal Chemistry Letters     ISSN:1948-5875  Volume:2  Issue:10  Page:774-779  

Burger Matthew T;   Pecchi Sabina;   Wagman Allan;   Ni Zhi-Jie;   Knapp Mark;   ...

来源数据库:[Web of Science, Science Citation Index Expanded, Scopus]         被引频次:112

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11    
Discovery of TAK-875: A potent, selective, and orally bioavailable GPR40 agonist 期刊论文

ACS Medicinal Chemistry Letters     ISSN:1948-5875  Volume:1  Issue:6  Page:290-294  

Negoro Nobuyuki;   Sasaki Shinobu;   Mikami Satoshi;   Ito Masahiro;   Suzuki Masami;   ...

来源数据库:[Web of Science, Science Citation Index Expanded, Scopus]         被引频次:161

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12    
Aminoindazole PDK1 inhibitors: A case study in fragment-based drug discovery 期刊论文

ACS Medicinal Chemistry Letters     ISSN:1948-5875  Volume:1  Issue:8  Page:439-442  

Medina Jesús R;   Blackledge Charles W;   Heerding Dirk A;   Campobasso Nino;   Ward Paris;   ...

来源数据库:[Web of Science, Science Citation Index Expanded, Scopus]         被引频次:20

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13    
Discovery of MK-5172, a macrocyclic hepatitis C virus NS3/4a protease inhibitor 期刊论文

ACS Medicinal Chemistry Letters     ISSN:1948-5875  Volume:3  Issue:4  Page:332-336  

Harper Steven;   McCauley John A;   Rudd Michael T;   Ferrara Marco;   DiFilippo Marcello;   ...

来源数据库:[Web of Science, Science Citation Index Expanded, Scopus]         被引频次:110

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14    
Discovery of NVP-LDE225, a potent and selective smoothened antagonist 期刊论文

ACS Medicinal Chemistry Letters     ISSN:1948-5875  Volume:1  Issue:3  Page:130-134  

Pan Shifeng;   Wu Xu;   Jiang Jiqing;   Gao Wenqi;   Wan Yongqin;   ...

来源数据库:[Web of Science, Science Citation Index Expanded, Scopus]         被引频次:142

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15    
Discovery of GSK2656157: An optimized PERK inhibitor selected for preclinical development 期刊论文

ACS Medicinal Chemistry Letters     ISSN:1948-5875  Volume:4  Issue:10  Page:964-968  

Axten Jeffrey M;   Romeril Stuart P;   Shu Arthur;   Ralph Jeffrey;   Medina Jesús R;   ...

来源数据库:[Web of Science, Science Citation Index Expanded, Scopus]         被引频次:75

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16    
Drawing the PDB: Protein-ligand complexes in two dimensions 期刊论文

ACS Medicinal Chemistry Letters     ISSN:1948-5875  Volume:1  Issue:9  Page:540-545  

Stierand Katrin;   Rarey Matthias;  

来源数据库:[Web of Science, Science Citation Index Expanded, Scopus]         被引频次:131

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17    
Discovery and development of potent and selective inhibitors of histone methyltransferase G9a 期刊论文

ACS Medicinal Chemistry Letters     ISSN:1948-5875  Volume:5  Issue:2  Page:205-209  

Sweis Ramzi F;   Pliushchev Marina;   Brown Peter J;   Guo Jun;   Li Fengling;   ...

来源数据库:[Web of Science, Science Citation Index Expanded, Scopus]         被引频次:69

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18    
Crystal structures and structure-activity relationships of imidazothiazole derivatives as IDO1 inhibitors 期刊论文

ACS Medicinal Chemistry Letters     ISSN:1948-5875  Volume:5  Issue:10  Page:1119-1123  

Tojo Shingo;   Kohno Tetsuya;   Tanaka Tomoyuki;   Kamioka Seiji;   Ota Yosuke;   ...

来源数据库:[Web of Science, Science Citation Index Expanded, Scopus]         被引频次:58

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19    
Discovery of AG-120 (Ivosidenib): A First-in-Class Mutant IDH1 Inhibitor for the Treatment of IDH1 Mutant Cancers 期刊论文

ACS Medicinal Chemistry Letters     ISSN:1948-5875  Volume:9  Issue:4  Page:300-305  

Popovici-Muller Janeta;   Lemieux René M;   Artin Erin;   Saunders Jeffrey O;   Salituro Francesco G;   ...

来源数据库:[Web of Science, Science Citation Index Expanded, Scopus]         被引频次:23

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20    
EPZ011989, A potent, orally-available EZH2 inhibitor with robust in vivo activity 期刊论文

ACS Medicinal Chemistry Letters     ISSN:1948-5875  Volume:6  Issue:5  Page:491-495  

Campbell John E;   Kuntz Kevin W;   Knutson Sarah K;   Warholic Natalie M;   Keilhack Heike;   ...

来源数据库:[Web of Science, Science Citation Index Expanded, Scopus]         被引频次:49

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